Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50035089
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093754((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)
Affinity DataIC50: 1.30E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093752((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)
Affinity DataIC50: 2.00E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093755((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)
Affinity DataIC50: 2.20E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 3.80E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093754((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)
Affinity DataIC50: 4.80E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093755((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)
Affinity DataIC50: 6.50E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 7.00E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 7.00E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093752((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)
Affinity DataIC50: 8.40E+3nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093754((2S, 3S)-3-Amino-2-(naphthalen-1-ylmethoxy)-pentan...)
Affinity DataIC50: 1.50E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093755((2S, 3S)-3-Amino-2-(naphthalen-2-ylmethoxy)-pentan...)
Affinity DataIC50: 1.60E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 2.10E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 2.30E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50247191((2S,3S)-2-Amino-3-benzyloxy-succinic acid | DL-thr...)
Affinity DataIC50: 4.80E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 6.40E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093752((2S, 3S)-3-Amino-2-methoxy-pentanedioic acid | CHE...)
Affinity DataIC50: 6.90E+4nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 1.61E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 3(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 1.61E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 2.21E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 2(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 2.21E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 6.37E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 6.37E+5nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetExcitatory amino acid transporter 1(Human)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50093753(DL-TBOA | (2S,3S)-2-amino-3-(benzyloxy)succinic ac...)
Affinity DataIC50: 1.00E+6nMAssay Description:Concentration required for blocking [14C]glutamate uptake in COS-1 cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed