Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50035092
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.0400nMAssay Description:Compound was evaluated for its ability to displace [3H]p-CI-DPDPE in C6 glioma cells expressing the cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  3.70nMAssay Description:Compound was evaluated for its ability to displace [3H]DAMGO in C6 glioma cells expressing the cloned Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  5.80nMAssay Description:Compound was evaluated for its ability to displace [3H]U-69593 in CHO cells expressing the cloned Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093785([1,5-3H]-17-Cyclohexylethyl-6,7-dehydro-4,5a -epox...)
Affinity DataKi:  7.30nMAssay Description:Compound was evaluated for its ability to displace [3H]DAMGO in C6 glioma cells expressing the cloned Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093784([1,5-3H]-17-Cyclohexylmethyl-6,7-dehydro-4,5a -epo...)
Affinity DataKi:  95nMAssay Description:Compound was evaluated for its ability to displace [3H]p-CI-DPDPE in C6 glioma cells expressing the cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093783([1,5-3H]-17-Benzyl-6,7-dehydro-4,5a -epoxy-3,14-di...)
Affinity DataKi:  115nMAssay Description:Compound was evaluated for its ability to displace [3H]p-CI-DPDPE in C6 glioma cells expressing the cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093783([1,5-3H]-17-Benzyl-6,7-dehydro-4,5a -epoxy-3,14-di...)
Affinity DataKi:  134nMAssay Description:Compound was evaluated for its ability to displace [3H]U-69593 in CHO cells expressing the cloned Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093785([1,5-3H]-17-Cyclohexylethyl-6,7-dehydro-4,5a -epox...)
Affinity DataKi:  181nMAssay Description:Compound was evaluated for its ability to displace [3H]p-CI-DPDPE in C6 glioma cells expressing the cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093785([1,5-3H]-17-Cyclohexylethyl-6,7-dehydro-4,5a -epox...)
Affinity DataKi:  378nMAssay Description:Compound was evaluated for its ability to displace [3H]U-69593 in CHO cells expressing the cloned Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093784([1,5-3H]-17-Cyclohexylmethyl-6,7-dehydro-4,5a -epo...)
Affinity DataKi:  1.12E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]U-69593 in CHO cells expressing the cloned Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093784([1,5-3H]-17-Cyclohexylmethyl-6,7-dehydro-4,5a -epo...)
Affinity DataKi:  1.93E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]DAMGO in C6 glioma cells expressing the cloned Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50093783([1,5-3H]-17-Benzyl-6,7-dehydro-4,5a -epoxy-3,14-di...)
Affinity DataKi:  5.33E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]DAMGO in C6 glioma cells expressing the cloned Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed