Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50010403
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094519((R)-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-phe...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094513(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-te...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094519((R)-3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-phe...)
Affinity DataIC50: 600nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094515(1,1,1-Trifluoro-3-{(3-phenoxy-phenyl)-[3-(1,1,2,2-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094525(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(4-trifluoro...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094524((R)-1,1,1-trifluoro-3-((3-(trifluoromethylthio)ben...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094513(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-te...)
Affinity DataIC50: 6.00E+3nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094516(3-((3-(trifluoromethoxy)benzyl)(3-fluorophenyl)ami...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094521(1,1,1-trifluoro-3-(phenyl(3-(trifluoromethyl)benzy...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094520(1,1,1-Trifluoro-3-[(3-fluoro-phenyl)-(4-trifluorom...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094515(1,1,1-Trifluoro-3-{(3-phenoxy-phenyl)-[3-(1,1,2,2-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094517(1,1,1-Trifluoro-3-[(4-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094518(1,1,1-Trifluoro-3-[(3-fluoro-phenyl)-(3-trifluorom...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50: 4.00E+4nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094522(1,1,1-Trifluoro-3-[(3-fluoro-phenyl)-(2-trifluorom...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094523(3-[Benzyl-(3-fluoro-phenyl)-amino]-1,1,1-trifluoro...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094526(1,1,1-trifluoro-3-((3-fluorophenyl)(3-methylbenzyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]CE from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094525(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(4-trifluoro...)
Affinity DataIC50: 1.20E+5nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094521(1,1,1-trifluoro-3-(phenyl(3-(trifluoromethyl)benzy...)
Affinity DataIC50: 2.00E+5nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094518(1,1,1-Trifluoro-3-[(3-fluoro-phenyl)-(3-trifluorom...)
Affinity DataIC50: 2.00E+5nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50094516(3-((3-(trifluoromethoxy)benzyl)(3-fluorophenyl)ami...)
Affinity DataIC50: 2.00E+5nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed