Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50035099
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095154((S)-2-[(S)-2-(2-{1-[(R)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity towards Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095154((S)-2-[(S)-2-(2-{1-[(R)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataIC50: 1.80nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 9.90nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095151((S)-2-[(S)-2-(2-{1-[(S)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataKi:  10nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095150(Endomorphin 1 | CHEMBL329996 | (R)-1-[(S)-2-Amino-...)
Affinity DataKi:  54nMAssay Description:Binding affinity towards Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 56nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095151((S)-2-[(S)-2-(2-{1-[(S)-2-Amino-3-((S)-4-hydroxy-p...)
Affinity DataIC50: 72nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095150(Endomorphin 1 | CHEMBL329996 | (R)-1-[(S)-2-Amino-...)
Affinity DataIC50: 470nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095152((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50: 680nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095152((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  908nMAssay Description:Binding affinity towards Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095156((S)-1-[3-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095157(1-[(R)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration required for inhibition of [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed