Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50048513
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219243(CHEMBL351300)
Affinity DataKi:  3.20nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219204(CHEMBL161916)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219202(CHEMBL161126)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50370572(SB-277011 | CHEMBL85606)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219203(CHEMBL161853)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219205(CHEMBL162193)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219250(CHEMBL160998)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219201(CHEMBL351722)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219243(CHEMBL351300)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219204(CHEMBL161916)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219202(CHEMBL161126)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219205(CHEMBL162193)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50370572(SB-277011 | CHEMBL85606)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <1.00E+3nMAssay Description:Evaluated for the binding affinity to 5-HT 2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219203(CHEMBL161853)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi:  1.26E+3nMAssay Description:Evaluated for the binding affinity against 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219201(CHEMBL351722)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219250(CHEMBL160998)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [125I]iodosulpiride from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi:  3.16E+3nMAssay Description:Evaluated for the binding affinity to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <3.98E+3nMAssay Description:Evaluated for the binding affinity to 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi:  5.01E+3nMAssay Description:Evaluated for the binding affinity to 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <5.01E+3nMAssay Description:Evaluated for the binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <5.01E+3nMAssay Description:Evaluated for the binding affinity to alpha 1B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <7.94E+3nMAssay Description:Evaluated for the binding affinity to 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50219200(CHEMBL158627)
Affinity DataKi: <1.00E+4nMAssay Description:Evaluated for the binding affinity towards 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details Article
PubMed