Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50035197
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50000041((+/-)(2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-...)
Affinity DataIC50: 2.90nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097740(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 410nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097732(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 510nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 980nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.67E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.67E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097726(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097740(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 2.31E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097730(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 2.43E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097742(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 3.60E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097743(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097738(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097731(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097725(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 7.93E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 7.93E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097728(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097723(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097734(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 2.40E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097729(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 2.40E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097737(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097736(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 4.60E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rabbit whole brain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097723(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097742(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097734(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097731(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097726(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097738(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097743(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rabbit whole brain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097729(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097725(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097728(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097730(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097732(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097737(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097736(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
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