Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50010705
LigandPNGBDBM50067584(2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bipheny...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50: 1nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097809((S)-2-[(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmet...)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50: 20nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097817((S)-2-({5-[(3-Cyclohexylmethyl-3H-imidazol-4-ylmet...)
Affinity DataIC50: 41nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50: 200nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097813(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 220nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097810((S)-2-({5-[(3-Biphenyl-4-ylmethyl-3H-imidazol-4-yl...)
Affinity DataIC50: 260nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097811(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 380nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097812(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 640nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097815((S)-2-({5-[(1-Cyclohexylmethyl-1H-imidazol-4-ylmet...)
Affinity DataIC50: 780nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50067584(2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bipheny...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097808((S)-4-Methylsulfanyl-2-({5-[(1-naphthalen-1-ylmeth...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097816(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097809((S)-2-[(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmet...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097818((S)-2-({5-[(1-Biphenyl-4-ylmethyl-1H-imidazol-4-yl...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097813(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097818((S)-2-({5-[(1-Biphenyl-4-ylmethyl-1H-imidazol-4-yl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097816(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097811(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097808((S)-4-Methylsulfanyl-2-({5-[(1-naphthalen-1-ylmeth...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097810((S)-2-({5-[(3-Biphenyl-4-ylmethyl-3H-imidazol-4-yl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed