Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010728
TargetD(2) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 220nMAssay Description:Inhibition of binding of [3H]spiroperidol to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 430nMAssay Description:Inhibition of binding of [3H]SCH-23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50: 450nMAssay Description:Inhibition of binding of [3H]SCH-23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50028970(6-Amino-5,6,7,8-tetrahydro-naphthalene-1,2-diol | ...)
Affinity DataIC50: 700nMAssay Description:Inhibition of binding of [3H]spiroperidol to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of binding of [3H]SCH-23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50219332(CHEMBL133432)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50219332(CHEMBL133432)
Affinity DataIC50: 6.75E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50219331(1,2,3,4,4A,5,10,10A-Octahydro-Benzo[G]Quinoline | ...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50: 2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50: 2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50: 6.67E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50: 6.67E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed