Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010815
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 7nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 27nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099028(1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099017(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 36nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099025(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099022(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 47nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099024(1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 48nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human Gonadotropin-releasing hormone receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099021(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099029(Ethanesulfonic acid [4-(4-{2-[2-(3,5-dimethyl-phen...)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099020(Propane-2-sulfonic acid [4-(4-{2-[2-(3,5-dimethyl-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099026({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099027(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099019(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 357nMAssay Description:Inhibition of human Gonadotropin-releasing hormone receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099018({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed