Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50035126
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099875((E)-2-Amino-5-(2,4-difluoro-phenyl)-5-(4-isopropyl...)
Affinity DataIC50: 150nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099886((E)-2-Amino-5-(3,4-diethyl-phenyl)-5-(2,4-difluoro...)
Affinity DataIC50: 283nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099859(Sodium; (E)-2-amino-5-(2-fluoro-phenyl)-5-(4-isopr...)
Affinity DataIC50: 290nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099862(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-i...)
Affinity DataIC50: 330nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099878((E)-2-Amino-5-(2,4-difluoro-phenyl)-5-naphthalen-2...)
Affinity DataIC50: 365nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099882(Sodium; (Z)-2-amino-5-(4-isopropyl-phenyl)-5-pheny...)
Affinity DataIC50: 400nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099879(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-e...)
Affinity DataIC50: 460nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099866(Sodium; (E)-2-amino-5-(3,4-diethyl-phenyl)-5-(2,4-...)
Affinity DataIC50: 660nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099883(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-naph...)
Affinity DataIC50: 770nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099858(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-thiop...)
Affinity DataIC50: 1.03E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099873(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-(4-me...)
Affinity DataIC50: 1.16E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099863(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-p-to...)
Affinity DataIC50: 1.17E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099868(Sodium; (E)-2-amino-5-biphenyl-3-yl-5-(2,4-difluor...)
Affinity DataIC50: 1.34E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099861(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-(3-i...)
Affinity DataIC50: 1.59E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099881((E)-2-Amino-5-(4-tert-butyl-phenyl)-5-(2,4-difluor...)
Affinity DataIC50: 1.74E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099865(Sodium; 2-amino-5,5-bis-(4-isopropyl-phenyl)-pent-...)
Affinity DataIC50: 2.03E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099880(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-m...)
Affinity DataIC50: 2.03E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099885(Sodium; (E)-2-amino-5-biphenyl-4-yl-5-(4-isopropyl...)
Affinity DataIC50: 2.06E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099864(Sodium; (Z)-2-amino-5-biphenyl-4-yl-5-(2,4-difluor...)
Affinity DataIC50: 2.40E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099872(Sodium; (E)-2-amino-5-(4-cyano-phenyl)-5-(4-isopro...)
Affinity DataIC50: 2.64E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099870(Sodium; (E)-2-amino-5-biphenyl-2-yl-5-(2,4-difluor...)
Affinity DataIC50: 2.75E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099864(Sodium; (Z)-2-amino-5-biphenyl-4-yl-5-(2,4-difluor...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099877(Sodium; (E)-2-amino-5-biphenyl-4-yl-5-(2,4-difluor...)
Affinity DataIC50: 3.66E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099871(Sodium; (E)-2-amino-5-(4-tert-butyl-phenyl)-5-(4-i...)
Affinity DataIC50: 5.47E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099858(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-thiop...)
Affinity DataIC50: 5.77E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099874(Sodium; (Z)-2-amino-5-(2,4-difluoro-phenyl)-5-thio...)
Affinity DataIC50: 5.88E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099867(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-pyrid...)
Affinity DataIC50: 5.93E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099884(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-phen...)
Affinity DataIC50: 6.44E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099867(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-pyrid...)
Affinity DataIC50: 6.48E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099859(Sodium; (E)-2-amino-5-(2-fluoro-phenyl)-5-(4-isopr...)
Affinity DataIC50: 8.02E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099882(Sodium; (Z)-2-amino-5-(4-isopropyl-phenyl)-5-pheny...)
Affinity DataIC50: 8.34E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099870(Sodium; (E)-2-amino-5-biphenyl-2-yl-5-(2,4-difluor...)
Affinity DataIC50: 8.92E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099884(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-phen...)
Affinity DataIC50: 9.50E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099863(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-p-to...)
Affinity DataIC50: 9.56E+3nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099877(Sodium; (E)-2-amino-5-biphenyl-4-yl-5-(2,4-difluor...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099872(Sodium; (E)-2-amino-5-(4-cyano-phenyl)-5-(4-isopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099860(Sodium; (Z)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-i...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099866(Sodium; (E)-2-amino-5-(3,4-diethyl-phenyl)-5-(2,4-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099881((E)-2-Amino-5-(4-tert-butyl-phenyl)-5-(2,4-difluor...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099869((E)-2-Amino-5-(2,4-difluoro-phenyl)-5-pyridin-3-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099883(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-naph...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099860(Sodium; (Z)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-i...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099868(Sodium; (E)-2-amino-5-biphenyl-3-yl-5-(2,4-difluor...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099869((E)-2-Amino-5-(2,4-difluoro-phenyl)-5-pyridin-3-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099885(Sodium; (E)-2-amino-5-biphenyl-4-yl-5-(4-isopropyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099873(Sodium; (E)-2-amino-5-(4-isopropyl-phenyl)-5-(4-me...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099876(Sodium; (E)-2-amino-5-(4-cyano-phenyl)-5-(2,4-difl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-2 (GlyT-2) transporter cells after incubation at 30 degrees for 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099865(Sodium; 2-amino-5,5-bis-(4-isopropyl-phenyl)-pent-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099876(Sodium; (E)-2-amino-5-(4-cyano-phenyl)-5-(2,4-difl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 1(Rat)
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50099879(Sodium; (E)-2-amino-5-(2,4-difluoro-phenyl)-5-(4-e...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro glycine reuptake inhibitory activity against glycine transporter type-1 isoform C (GlyT-1c) transporter cells after incubation at 30 degrees...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
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