Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50010944
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100403({3-[4-(4-Bromo-phenyl)-thiazol-2-ylmethyl]-5-metho...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100395([3-(4-Benzo[b]thiophen-3-yl-thiazol-2-ylmethyl)-5-...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100400((4-Bromo-phenyl)-{5-methoxy-2-methyl-3-[4-(4-nitro...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100401((4-Bromo-phenyl)-{3-[4-(4-chloro-phenyl)-thiazol-2...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100404((4-Chloro-phenyl)-[5-methoxy-2-methyl-3-(4-naphtha...)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100396({3-[4-(3-Bromo-phenyl)-thiazol-2-ylmethyl]-5-metho...)
Affinity DataIC50: 8nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100399((4-Chloro-phenyl)-{3-[4-(4-fluoro-phenyl)-thiazol-...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100402((4-Chloro-phenyl)-{5-methoxy-2-methyl-3-[4-(4-nitr...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100397((4-Chloro-phenyl)-{3-[4-(4-chloro-phenyl)-thiazol-...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100405((4-Bromo-phenyl)-{3-[4-(4-bromo-phenyl)-thiazol-2-...)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100398(4-{2-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100394([3-(2-Amino-thiazol-4-ylmethyl)-5-methoxy-2-methyl...)
Affinity DataIC50: 390nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 2 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 1 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50100394([3-(2-Amino-thiazol-4-ylmethyl)-5-methoxy-2-methyl...)
Affinity DataIC50: 1.55E+7nMAssay Description:Inhibitory concentration against human recombinant Prostaglandin G/H synthase 1 cloned and expressed in baculovirus (Sf9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed