Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50010990
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50094513(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(1,1,2,2-te...)
Affinity DataIC50: 200nMAssay Description:In vitro human CETP inhibitory activity was assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(furan-2-yl...)
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101002(3-((4-fluoro-3-(furan-2-yl)benzyl)(3-phenoxyphenyl...)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100996(1,1,1-Trifluoro-3-[(3-furan-3-yl-benzyl)-(3-phenox...)
Affinity DataIC50: 910nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100999(3-((3-(thiophen-2-yl)benzyl)(3-phenoxyphenyl)amino...)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101008(3-((3-(furan-2-yl)-4-methylbenzyl)(3-phenoxyphenyl...)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101007(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(3-(trifluo...)
Affinity DataIC50: 4.08E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101000(3-((biphenyl-3-ylmethyl)(3-phenoxyphenyl)amino)-1,...)
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101003(3-((3-ethoxybenzyl)(3-phenoxyphenyl)amino)-1,1,1-t...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor par...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101006(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-pyridin-4...)
Affinity DataIC50: 6.24E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100998(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(pyrimidin-...)
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101009(1,1,1-Trifluoro-3-[[3-(1-methyl-1H-pyrrol-2-yl)-be...)
Affinity DataIC50: 6.79E+3nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101001(3-((3-(pyridin-3-yl)benzyl)(3-phenoxyphenyl)amino)...)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101005(1,1,1-trifluoro-3-((3-(3-methylpyridin-2-yl)benzyl...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101010(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-pyridin-2...)
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101004(1,1,1-trifluoro-3-((3-(furan-2-yl)-4-morpholinoben...)
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101000(3-((biphenyl-3-ylmethyl)(3-phenoxyphenyl)amino)-1,...)
Affinity DataIC50: 4.70E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor par...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101002(3-((4-fluoro-3-(furan-2-yl)benzyl)(3-phenoxyphenyl...)
Affinity DataIC50: 4.90E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor par...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-trifluoro-3-((3-phenoxyphenyl)(3-(furan-2-yl...)
Affinity DataIC50: 5.20E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor par...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50100999(3-((3-(thiophen-2-yl)benzyl)(3-phenoxyphenyl)amino...)
Affinity DataIC50: 8.30E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]cholesteryl ester ([3H]CE) from HDL donor particles to LDL acceptor par...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed