Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50035135
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50001023((2R,6R,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  0.310nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50001023((2R,6R,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity towards guinea pig Opioid receptor mu 1 using radioligand [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101160(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards guinea pig Opioid receptor mu 1 using radioligand [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101160(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  0.880nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50128411(4-cyclopropylmethyl-17-hydroxy-14-oxo-(1S,5R,13R,1...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50128411(4-cyclopropylmethyl-17-hydroxy-14-oxo-(1S,5R,13R,1...)
Affinity DataKi:  22nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  24nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101158(14-hydroxy-4-methyl-(1S,5R,17R)-12-oxa-4-azapentac...)
Affinity DataKi:  34nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50128411(4-cyclopropylmethyl-17-hydroxy-14-oxo-(1S,5R,13R,1...)
Affinity DataKi:  110nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101162(4,10N-dimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-4-aza...)
Affinity DataKi:  440nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101158(14-hydroxy-4-methyl-(1S,5R,17R)-12-oxa-4-azapentac...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101158(14-hydroxy-4-methyl-(1S,5R,17R)-12-oxa-4-azapentac...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101159(4,10N,10N-trimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-...)
Affinity DataKi:  5.80E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 of guinea pig brain membranes using radioligand 0.25 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101162(4,10N-dimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-4-aza...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101159(4,10N,10N-trimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U69,593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101162(4,10N-dimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-4-aza...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101159(4,10N,10N-trimethyl-14-hydroxy-(1S,5R,17R)-12-oxa-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards guinea pig Opioid receptor kappa 1 using radioligand [3H]U-69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed