Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 5322
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85212(CAS_5311260 | NSC_5311260 | LY341495)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50074749(LY379268 | (1R,4R,5S,6R)-4-Amino-2-oxa-bicyclo[3.1...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50034503(DCG-IV | (2S,2'R,3'R)-2-(2',3')-dicarboxycycloprop...)
Affinity DataKi:  61nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50013055(glutamic acid dianion | 2-aminopentanedioateglutam...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50004899(L-CCG-IV | 2-(Amino-carboxy-methyl)-cyclopropaneca...)
Affinity DataKi:  334nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50049747(LY307452 | CHEMBL166775 | (2S,4R)-2-Amino-4-(4,4-d...)
Affinity DataKi:  2.01E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50052398(2R, 4R-APDC | (2R,4R)-APDC | CHEMBL40086 | (2R,4R)...)
Affinity DataKi:  2.73E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85017((1S,3S)-HOMO-ACPD | (1S,3S)-1-AMINO-1-CARBOXYCYCLO...)
Affinity DataKi:  8.69E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85211(t-PDC | t-2,4-PDC)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50004881(Amino-(4-phosphono-phenyl)-acetic acid(RS-PPG) | (...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM17660(2-amino-3-(3,5-dioxo[1,2,4]oxadiazolidin-2-yl)prop...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM17658([3H]NAAG | (2S)-2-[(3S)-3-acetamido-3-formamidopro...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50089910(CHEMBL86508 | MPPG | 2-Amino-2-(4-phosphono-phenyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50030627(CHEMBL299683 | MCPG | (R,S)-alpha-Methyl-4-carboxy...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50056272((2S,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxy...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM18125(L-Aspartic acid, 2 | L-Aspartate | CHEMBL274323 | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50004051(CHEMBL285843 | 2-Amino-4-phosphono-butyric acid | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85077(CAS_23052-80-4 | NSC_3857 | 3-Phosphono-D,L-2-amin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM85707(CAS_82410-32-0 | NSC_3454 | DHPG)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50327886(CHEMBL1256243 | Anti-endo-MPDC | (1R,2S,5S,6S)-3-a...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetGlutamate receptor 3(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50004863(1S, 3R-ACPD | CHEMBL29726 | 1R,3R-ACPD | 1R,3S-ACP...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed