Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50011065
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101892(2-(7-Ethoxy-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50: 40nMAssay Description:Compound was evaluated for its ability to inhibit human Purinergic receptor P2Y12 expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101903(N-(6-Ethoxy-benzothiazol-2-yl)-2-(6-ethoxy-benzoth...)
Affinity DataIC50: 170nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101892(2-(7-Ethoxy-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50: 170nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101894(2-(4-Hydroxy-7-methoxy-2,2-dioxo-2H-2lambda*6*,9-d...)
Affinity DataIC50: 800nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101898(2-(4-Hydroxy-7-methanesulfonyl-2,2-dioxo-2H-2lambd...)
Affinity DataIC50: 1.10E+3nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101896(3-[2-(6-Ethoxycarbonyl-benzothiazol-2-ylsulfamoyl)...)
Affinity DataIC50: 1.80E+3nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101890(2-(4-Hydroxy-2,2-dioxo-2H-2lambda*6*,9-dithia-1,4a...)
Affinity DataIC50: 2.10E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101893(2-(4-Hydroxy-7-methyl-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50: 2.20E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101895(2-(7-Chloro-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50: 3.50E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101900(2-(4-Hydroxy-7-nitro-2,2-dioxo-2H-2lambda*6*,9-dit...)
Affinity DataIC50: 3.50E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101897(2-(7-Fluoro-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...)
Affinity DataIC50: 3.70E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101902(2-(4-Hydroxy-2,2-dioxo-7-phenyl-2H-2lambda*6*,9-di...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101899(2-(4-Hydroxy-2,2-dioxo-7-phenoxy-2H-2lambda*6*,9-d...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101891(5-Methoxy-2,2-dioxo-2H-2lambda*6*,9-dithia-1,4a-di...)
Affinity DataIC50: 7.70E+4nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101901(2,2-Dioxo-7-trifluoromethoxy-2H-2lambda*6*,9-dithi...)
Affinity DataIC50: 1.20E+5nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50101889(2-(7-Cyclohexyl-4-hydroxy-2,2-dioxo-2H-2lambda*6*,...)
Affinity DataIC50: 1.20E+5nMAssay Description:Ability to displace [3H]2-MeS-ADP from human Purinergic receptor P2Y12More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed