Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50011207
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103757((1S,2R,3S,4R,5S)-4-(1,3-Dibutyl-2,6-dioxo-1,2,3,6-...)
Affinity DataKi:  1.86E+3nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103755(1,3-Dibutyl-7-((1S,2R,3S,4R,5R)-3,4-dihydroxy-5-hy...)
Affinity DataKi: <2.97E+3nMAssay Description:Displacement of [3H]R-PIA binding to Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103755(1,3-Dibutyl-7-((1S,2R,3S,4R,5R)-3,4-dihydroxy-5-hy...)
Affinity DataKi:  4.35E+3nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103758((R)-Phosphoric acid mono-[(S)-(1S,3R,6R)-2,3-dihyd...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103753((2R,4S)-4-(2-Amino-6-hydroxy-purin-9-yl)-1-((R)-(R...)
Affinity DataKi:  2.05E+4nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103756(dimer[Phosphoric acid mono-[(1R,2R,3S,4R,5S)-2,3-d...)
Affinity DataKi:  2.16E+4nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103757((1S,2R,3S,4R,5S)-4-(1,3-Dibutyl-2,6-dioxo-1,2,3,6-...)
Affinity DataKi: <2.44E+4nMAssay Description:Displacement of [3H]R-PIA binding to Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103754((1S,2R,6S)-2,3-Dihydroxy-4-(6-hydroxy-purin-9-yl)-...)
Affinity DataKi:  2.88E+4nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50103752((1S,2R,3R,6R)-1-((S)-Hydroxymethyl)-4-(6-hydroxy-p...)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed