Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50011280
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50101321([(S)-1-((S)-1-Benzyl-2-benzyloxycarbamoyl-2-oxo-et...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104576([(S)-1-((S)-1-Benzyl-2-methoxycarbamoyl-2-oxo-ethy...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104586([(R)-1-((S)-1-Benzyl-2-benzyloxycarbamoyl-2-oxo-et...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104579({(S)-1-[(S)-1-((S)-1-Benzyl-2-benzyloxycarbamoyl-2...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104587([(S)-1-((S)-1-Benzyl-2-oxo-2-pentafluorophenylmeth...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50101317([(S)-1-((S)-1-Benzyl-2-ethoxycarbamoyl-2-oxo-ethyl...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104585({(S)-1-[(S)-1-((S)-1-Benzyl-2-methoxycarbamoyl-2-o...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104577({(S)-1-[(S)-1-Benzyl-2-(4-methyl-cyclohexyloxycarb...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104581([(S)-1-((S)-1-Benzyloxyaminooxalyl-pentylcarbamoyl...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104584([(S)-1-((S)-1-Benzyl-2-tert-butoxycarbamoyl-2-oxo-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104583((S)-N-Benzyloxy-3-((R)-3-benzyloxy-2-methanesulfon...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104582((R)-N-((S)-1-Benzylcarbamoyl-2-phenyl-ethyl)-3-ben...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104578((R)-3-Benzyloxy-N-((S)-1-ethylcarbamoyl-2-phenyl-e...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104580((S)-3-((R)-3-Benzyloxy-2-methanesulfonylamino-prop...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104589((S)-N-Benzyloxy-3-((R)-3-benzyloxy-2-methanesulfon...)
Affinity DataIC50: 152nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50104588(N-[(S)-1-((S)-1-Ethoxyaminooxalyl-pentylcarbamoyl)...)
Affinity DataIC50: 193nMAssay Description:Inhibition of human recombinant Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed