Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50011286
TargetCalpain-1 catalytic subunit(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50104647((3S,6S)-3,6-Bis-(4-hydroxy-benzyl)-1,4-dimethyl-pi...)
Affinity DataIC50: 800nMAssay Description:Compound was tested for its inhibitory activity against calpain isolated from Streptomyces speciesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50104646(6-Benzyl-3-isopropyl-1H-pyrazin-2-one | CHEMBL4194...)
Affinity DataIC50: 1.20E+3nMAssay Description:Compound was tested for its inhibitory activity against calpain isolated from Streptomyces speciesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed