Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003588
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382379(CHEMBL420134)
Affinity DataIC50: 36nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382370(CHEMBL326629)
Affinity DataIC50: 100nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382380(CHEMBL115491)
Affinity DataIC50: 180nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382357(CHEMBL326089)
Affinity DataIC50: 200nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382358(CHEMBL324091)
Affinity DataIC50: 220nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382369(CHEMBL113806)
Affinity DataIC50: 250nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50473403(CHEMBL326591)
Affinity DataIC50: 250nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382381(CHEMBL331361)
Affinity DataIC50: 265nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382372(CHEMBL114430)
Affinity DataIC50: 280nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382375(CHEMBL117211)
Affinity DataIC50: 360nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382371(CHEMBL114962)
Affinity DataIC50: 450nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382378(CHEMBL431865)
Affinity DataIC50: 500nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382376(CHEMBL114057)
Affinity DataIC50: 800nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382356(CHEMBL114121)
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382373(CHEMBL324089)
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50382377(CHEMBL326944)
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity against p38 MAP kinase systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed