Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50036974
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105262(2-{3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-2-biphe...)
Affinity DataKi:  1.20nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataKi:  1.70nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105263(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  2nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105261(benzyl 2-[(2S)-2-({[(2S)-2-azaniumyl-4-(methylsulf...)
Affinity DataKi:  2nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105262(2-{3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-2-biphe...)
Affinity DataKi:  2.90nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105263(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  4.80nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105261(benzyl 2-[(2S)-2-({[(2S)-2-azaniumyl-4-(methylsulf...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataKi:  7.00E+3nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed