Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50011374
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105862(pGlu-His-Trp-Ser-Tyr-D-Lys(2-(hydroxymethyl)anthra...)
Affinity DataIC50: 0.00200nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105860(pGlu-His-Trp-Ser-Tyr-D-Lys-Leu-Arg-Pro-Gly-NH2([D-...)
Affinity DataIC50: 0.0800nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105861(pGlu-His-Trp-Ser-Tyr-D-Lys(N-(2 chloro-1,4-naphtho...)
Affinity DataIC50: 0.0900nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50105863(pGlu-His-Trp-Ser-Tyr-D-Lys(emodic acid(1,6,8-trihy...)
Affinity DataIC50: 0.25nMAssay Description:Evaluated for gonadotropin-releasing hormone receptor binding by displacing the 50% of the bound tracer [125I][D-Lys6]-GnRH radioligand in rat pituit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed