Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50011397
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106107(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  81nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106108(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(3,4-...)
Affinity DataEC50:  710nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  620nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106107(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  620nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  4nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  28nMAssay Description:Agonist activity against PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106104(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106106(2-(3-{3-[(3,4-Bis-trifluoromethyl-benzoyl)-(2-cycl...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106109(4-Isocyanato-benzoic acid 2-((2,4-bis-trifluoromet...)
Affinity DataEC50:  230nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity against PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106104(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  170nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106109(4-Isocyanato-benzoic acid 2-((2,4-bis-trifluoromet...)
Affinity DataEC50:  0.5nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106109(4-Isocyanato-benzoic acid 2-((2,4-bis-trifluoromet...)
Affinity DataEC50:  160nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106106(2-(3-{3-[(3,4-Bis-trifluoromethyl-benzoyl)-(2-cycl...)
Affinity DataEC50:  59nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106108(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(3,4-...)
Affinity DataEC50:  30nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106108(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(3,4-...)
Affinity DataEC50:  93nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106107(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  430nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR delta chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106106(2-(3-{3-[(3,4-Bis-trifluoromethyl-benzoyl)-(2-cycl...)
Affinity DataEC50:  320nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR gamma chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonist activity against PPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50106104(2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-ph...)
Affinity DataEC50:  230nMAssay Description:Agonistic transcriptional activity in CV-1 cells expressing Gal4-PPAR alpha chimeraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed