Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50003591
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 386nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 603nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 644nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 672nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 750nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 759nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 851nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 853nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.45E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 1.93E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 2.39E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florence
Curated by ChEMBL
University of Florence
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair








































