Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50011427
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106476(FGGFTGCRKSCRK | CHEMBL435511)
Affinity DataEC50:  156nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106472(CFGGFTCARKSARK | CHEMBL405451)
Affinity DataEC50: >1.00E+4nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataEC50:  1.12nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106481(CFGGFTGARKCARK | CHEMBL406010)
Affinity DataEC50:  439nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106469(FGGFTCARKCARK | cyclo[Cys6,Cys10]N/OFQ(1-13)NH2 | ...)
Affinity DataEC50:  31.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106478(FGGFTGARKCARKC | CHEMBL443591)
Affinity DataEC50:  4.37nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106475(FGGFTGCRKSCRK | CHEMBL266667)
Affinity DataEC50:  26.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106474(CFGGFTGARKCARK | CHEMBL405948)
Affinity DataEC50:  286nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106477(FGGFTGARKSARKLADE | Phe-GGFTGARKSARKLAD-Glu | CHEM...)
Affinity DataEC50:  1.93nMAssay Description:Binding of compound to cell membranes expressing human ORL1 receptor in HEk-293 cells using [32S]GTP-gamma-SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106467(FGGFTGCRKSARKC | CHEMBL384866)
Affinity DataEC50:  22.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106471(FGGFTGARKCARKC | CHEMBL406718)
Affinity DataEC50:  3.90nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106480(FGGFTGARKSARKL | CHEMBL437915)
Affinity DataEC50:  1.97nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106468(FGGFTGCRKSARKC | CHEMBL424934)
Affinity DataEC50:  25nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106470(FGGFTCARKCARK | CHEMBL442113)
Affinity DataEC50:  29.7nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106473(CFGGFTCARKSARK | CHEMBL268145)
Affinity DataEC50: >1.00E+4nMAssay Description:Efficacy for human ORL1 receptor expressing HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106478(FGGFTGARKCARKC | CHEMBL443591)
Affinity DataIC50: 0.122nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106477(FGGFTGARKSARKLADE | Phe-GGFTGARKSARKLAD-Glu | CHEM...)
Affinity DataIC50: 0.286nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106479(FGGFTGARKSARK | H-FGGFTGARKSARK-NH2 | NC(1-13)NH2 ...)
Affinity DataIC50: 0.353nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106471(FGGFTGARKCARKC | CHEMBL406718)
Affinity DataIC50: 0.471nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106480(FGGFTGARKSARKL | CHEMBL437915)
Affinity DataIC50: 0.520nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106469(FGGFTCARKCARK | cyclo[Cys6,Cys10]N/OFQ(1-13)NH2 | ...)
Affinity DataIC50: 0.833nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106470(FGGFTCARKCARK | CHEMBL442113)
Affinity DataIC50: 3.03nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106476(FGGFTGCRKSCRK | CHEMBL435511)
Affinity DataIC50: 3.04nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106468(FGGFTGCRKSARKC | CHEMBL424934)
Affinity DataIC50: 4.97nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106475(FGGFTGCRKSCRK | CHEMBL266667)
Affinity DataIC50: 8.70nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106467(FGGFTGCRKSARKC | CHEMBL384866)
Affinity DataIC50: 37.2nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106481(CFGGFTGARKCARK | CHEMBL406010)
Affinity DataIC50: 387nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106472(CFGGFTCARKSARK | CHEMBL405451)
Affinity DataIC50: 874nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106474(CFGGFTGARKCARK | CHEMBL405948)
Affinity DataIC50: 1.29E+3nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106473(CFGGFTCARKSARK | CHEMBL268145)
Affinity DataIC50: 2.71E+3nMAssay Description:Displacement of [3H]NC from human ORL1 receptor expressing HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed