Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50011582
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108309(2-(3H-Benzo[e]indol-1-yl)-1-methyl-ethylamine | CH...)
Affinity DataKi:  3nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  3.80nMAssay Description:Tested for binding affinity towards human 5-hydroxytryptamine 2C receptor using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  3.90nMAssay Description:Tested for binding affinity towards human 5-hydroxytryptamine 2C receptor using [3H]DOB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108309(2-(3H-Benzo[e]indol-1-yl)-1-methyl-ethylamine | CH...)
Affinity DataKi:  9nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  12nMAssay Description:Tested for binding affinity towards human 5-hydroxytryptamine 2A receptor using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  15nMAssay Description:Tested for binding affinity towards rat 5-hydroxytryptamine 2A receptor using [3H]DOB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108312(2-Benzo[g]indol-1-yl-1-methyl-ethylamine | CHEMBL3...)
Affinity DataKi:  38nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  39nMAssay Description:Tested for binding affinity towards human 5-hydroxytryptamine 2A receptor using [3H]DOB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108312(2-Benzo[g]indol-1-yl-1-methyl-ethylamine | CHEMBL3...)
Affinity DataKi:  42nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108315(7-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108314(8-Chloro-10-methoxy-1,2,3,4-tetrahydro-pyrazino[1,...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108315(7-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  85nMAssay Description:Tested for binding affinity towards human 5-hydroxytryptamine 2C receptor using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  85nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108314(8-Chloro-10-methoxy-1,2,3,4-tetrahydro-pyrazino[1,...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108317([2-(5,6-Difluoro-indol-1-yl)-ethyl]-dimethyl-amine...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108317([2-(5,6-Difluoro-indol-1-yl)-ethyl]-dimethyl-amine...)
Affinity DataKi:  300nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108318(6-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108306((S)-2-(5,6-Difluoro-indol-1-yl)-1-methyl-ethylamin...)
Affinity DataKi:  320nMAssay Description:Tested for binding affinity towards rat 5-hydroxytryptamine 2A receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108304(8-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108303(6-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108314(8-Chloro-10-methoxy-1,2,3,4-tetrahydro-pyrazino[1,...)
Affinity DataKi:  330nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108310(8-Chloro-10-methyl-1,2,3,4-tetrahydro-pyrazino[1,2...)
Affinity DataKi:  450nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108320([2-(6-Methoxy-indol-1-yl)-ethyl]-dimethyl-amine | ...)
Affinity DataKi:  490nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108303(6-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  520nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108315(7-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  560nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108308((2-Indol-1-yl-ethyl)-dimethyl-amine | (2-Indol-1-y...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108303(6-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108307(1,2,3,4-Tetrahydro-pyrazino[1,2-a]indole | CHEMBL6...)
Affinity DataKi:  635nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108317([2-(5,6-Difluoro-indol-1-yl)-ethyl]-dimethyl-amine...)
Affinity DataKi:  640nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108308((2-Indol-1-yl-ethyl)-dimethyl-amine | (2-Indol-1-y...)
Affinity DataKi:  650nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108308((2-Indol-1-yl-ethyl)-dimethyl-amine | (2-Indol-1-y...)
Affinity DataKi:  720nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108316(8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108318(6-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108320([2-(6-Methoxy-indol-1-yl)-ethyl]-dimethyl-amine | ...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108307(1,2,3,4-Tetrahydro-pyrazino[1,2-a]indole | CHEMBL6...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108310(8-Chloro-10-methyl-1,2,3,4-tetrahydro-pyrazino[1,2...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108311(7-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  1.30E+3nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108304(8-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  1.46E+3nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108304(8-Chloro-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole ...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108318(6-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  1.99E+3nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108319(2-Benzo[g]indol-1-yl-propylamine | CHEMBL42923)
Affinity DataKi:  4.30E+3nMAssay Description:Tested for binding affinity towards 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108307(1,2,3,4-Tetrahydro-pyrazino[1,2-a]indole | CHEMBL6...)
Affinity DataKi:  4.78E+3nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108311(7-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  5.16E+3nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108311(7-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  5.19E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108316(8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  5.83E+3nMAssay Description:Displacement of [3H]ketanserin from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108316(8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  9.93E+3nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108319(2-Benzo[g]indol-1-yl-propylamine | CHEMBL42923)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108313([2-(5-Methoxy-indol-1-yl)-ethyl]-dimethyl-amine | ...)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for binding affinity towards 5-HT2c receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108305(1,2,3,4-Tetrahydro-benzo[4,5]imidazo[1,2-a]pyrazin...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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