Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50035252
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108490((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 0.110nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108487((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108487((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 0.440nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108490((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 0.540nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50366797(CHEMBL1790503)
Affinity DataIC50: 1.10nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108486((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 1.40nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108489((3R,6S,9S)-9-(2-Amino-ethyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 3.5nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108486((3R,6S,9S)-9-(4-Amino-butyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 6.20nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50366797(CHEMBL1790503)
Affinity DataIC50: 6.30nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108491((3S,6R,9S)-3-(2-Amino-ethyl)-4-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 21nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108489((3R,6S,9S)-9-(2-Amino-ethyl)-1-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 40nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108488({(2R,5S,8S)-5-(4-Amino-butyl)-4-[(S)-2-amino-3-(4-...)
Affinity DataIC50: 74nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108488({(2R,5S,8S)-5-(4-Amino-butyl)-4-[(S)-2-amino-3-(4-...)
Affinity DataIC50: 79nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the guinea pig ileum mediated through mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50108491((3S,6R,9S)-3-(2-Amino-ethyl)-4-[(S)-2-amino-3-(4-h...)
Affinity DataIC50: 252nMAssay Description:Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed