Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011636
TargetThyroid hormone receptor beta(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108809([2,6-Diiodo-4-(2-methyl-benzofuran-3-carbonyl)-phe...)
Affinity DataIC50: 480nMAssay Description:Concentration required to inhibit 50% of binding of [125I]T3 to human Thyroid hormone receptor beta 1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM18957((2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-di...)
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit 50% of binding of [125I]T3 to human Thyroid hormone receptor beta 1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM18957((2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-di...)
Affinity DataIC50: 650nMAssay Description:Concentration required to inhibit 50% of binding of [125I]-T3 to human Thyroid hormone receptor alpha-1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108809([2,6-Diiodo-4-(2-methyl-benzofuran-3-carbonyl)-phe...)
Affinity DataIC50: 820nMAssay Description:Concentration required to inhibit 50% of binding of [125I]-T3 to human Thyroid hormone receptor alpha-1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108808([4-(2-Butyl-benzofuran-3-carbonyl)-2,6-diiodo-phen...)
Affinity DataIC50: 1.40E+3nMAssay Description:Concentration required to inhibit 50% of binding of [125I]-T3 to human Thyroid hormone receptor alpha-1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108808([4-(2-Butyl-benzofuran-3-carbonyl)-2,6-diiodo-phen...)
Affinity DataIC50: 4.00E+3nMAssay Description:Concentration required to inhibit 50% of binding of [125I]T3 to human Thyroid hormone receptor beta 1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108807([2,6-Diiodo-4-(2-methyl-benzofuran-3-ylmethyl)-phe...)
Affinity DataIC50: 4.50E+3nMAssay Description:Concentration required to inhibit 50% of binding of [125I]-T3 to human Thyroid hormone receptor alpha-1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50108807([2,6-Diiodo-4-(2-methyl-benzofuran-3-ylmethyl)-phe...)
Affinity DataIC50: 5.10E+3nMAssay Description:Concentration required to inhibit 50% of binding of [125I]T3 to human Thyroid hormone receptor beta 1 in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed