Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50037111
TargetMuscarinic acetylcholine receptor M3(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109647(Enablex | 2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-et...)
Affinity DataKi:  0.840nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109650(N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-ca...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109647(Enablex | 2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-et...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109644(N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109647(Enablex | 2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-et...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109647(Enablex | 2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-et...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109650(N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-ca...)
Affinity DataKi:  17nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS to membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109647(Enablex | 2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-et...)
Affinity DataKi:  47nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS to membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109650(N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-ca...)
Affinity DataKi:  60nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109644(N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(...)
Affinity DataKi:  74nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109650(N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-ca...)
Affinity DataKi:  77nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109650(N-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-ca...)
Affinity DataKi:  200nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109644(N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(...)
Affinity DataKi:  270nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS to membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109644(N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(...)
Affinity DataKi:  300nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109644(N-(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-4-[2-(...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity (Ki) against binding of [3H]NMS using membranes from CHO cells expressing cloned human Muscarinic acetylcholine receptor M5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed