Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50011839
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50088679(2-Phenyl-isoindole-1,3-dione | 2-phenylisoindoline...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50219329(CHEMBL8968)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066441(2-(2,6-Dimethyl-phenyl)-isoindole-1,3-dione | 2-(2...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50088679(2-Phenyl-isoindole-1,3-dione | 2-phenylisoindoline...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50219329(CHEMBL8968)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066441(2-(2,6-Dimethyl-phenyl)-isoindole-1,3-dione | 2-(2...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111216(5-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111221(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-4-nitro-...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111216(5-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111222(4-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111209(2-(2,3,5,6-Tetramethyl-phenyl)-isoindole-1,3-dione...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111217(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-isoindol...)
Affinity DataIC50: 290nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111213(2-(2,3,5-Trimethyl-phenyl)-isoindole-1,3-dione | C...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50070114(CHEMBL468 | 2-(2,6-dioxopiperidin-3-yl)isoindoline...)
Affinity DataIC50: 370nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111221(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-4-nitro-...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111220(2-(2,4-Dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl)-is...)
Affinity DataIC50: 440nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50070114(CHEMBL468 | 2-(2,6-dioxopiperidin-3-yl)isoindoline...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111211(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-5-nitro-...)
Affinity DataIC50: 540nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111207(2-(2,4-Dioxo-tetrahydro-pyrimidin-1-yl)-isoindole-...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111214(2-[2-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-eth...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111209(2-(2,3,5,6-Tetramethyl-phenyl)-isoindole-1,3-dione...)
Affinity DataIC50: 670nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111217(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-isoindol...)
Affinity DataIC50: 730nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111219(2-(2-Oxo-piperidin-3-yl)-isoindole-1,3-dione | CHE...)
Affinity DataIC50: 850nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111207(2-(2,4-Dioxo-tetrahydro-pyrimidin-1-yl)-isoindole-...)
Affinity DataIC50: 900nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111213(2-(2,3,5-Trimethyl-phenyl)-isoindole-1,3-dione | C...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111219(2-(2-Oxo-piperidin-3-yl)-isoindole-1,3-dione | CHE...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111214(2-[2-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-eth...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111211(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-5-nitro-...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111222(4-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111212(2-(4,6-Dimethoxy-pyrimidin-2-yl)-4H-isoquinoline-1...)
Affinity DataIC50: 3.57E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111220(2-(2,4-Dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl)-is...)
Affinity DataIC50: 3.81E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111224(2-(4,6-Dimethyl-pyrimidin-2-yl)-4H-isoquinoline-1,...)
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111208(2-(4,6-Dimethyl-pyridin-2-yl)-4H-isoquinoline-1,3-...)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111223(2-(3,5-Dimethyl-phenyl)-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111224(2-(4,6-Dimethyl-pyrimidin-2-yl)-4H-isoquinoline-1,...)
Affinity DataIC50: 8.33E+3nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111215(2-(4-Methoxy-6-methyl-pyrimidin-2-yl)-4H-isoquinol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111212(2-(4,6-Dimethoxy-pyrimidin-2-yl)-4H-isoquinoline-1...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111208(2-(4,6-Dimethyl-pyridin-2-yl)-4H-isoquinoline-1,3-...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111223(2-(3,5-Dimethyl-phenyl)-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111215(2-(4-Methoxy-6-methyl-pyrimidin-2-yl)-4H-isoquinol...)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111210(2-(3,5-Dimethyl-phenyl)-4H-isoquinoline-1,3-dione ...)
Affinity DataIC50: 3.85E+4nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111210(2-(3,5-Dimethyl-phenyl)-4H-isoquinoline-1,3-dione ...)
Affinity DataIC50: 9.52E+4nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed