Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50011943
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-azoni...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-azoni...)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  12.9nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  16.8nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  23nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  40nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  49nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  90nMAssay Description:Ability to displace [3H]WIN-35 radioligand for the dopamine transporter 428 DAT in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  133nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  133nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  269nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  269nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-azoni...)
Affinity DataKi:  610nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  642nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  642nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  690nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112329((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  690nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.02E+3nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.02E+3nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.86E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.89E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.04E+3nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.04E+3nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.23E+3nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.23E+3nMAssay Description:Ability to displace [3H]-nisoxatine radioligand for the Norepinephrine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.68E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  2.68E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-azoni...)
Affinity DataKi:  3.26E+3nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  3.74E+3nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  3.74E+3nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  4.38E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112328(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  4.38E+3nMAssay Description:Ability to displace [3H]pirenzepine radioligand for the Muscarinic acetylcholine receptor M1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50112327(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to displace [3H]citalopram radioligand, for the Serotonin transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed