Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50023759
TargetPlasmepsin II(Plasmodium falciparum)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250839(CHEMBL2058413 | CHEMBL511879 | 6-bromo-2'-de-N-met...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250839(CHEMBL2058413 | CHEMBL511879 | 6-bromo-2'-de-N-met...)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin-2 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]methylspiperone form human cloned 5HT2A receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250840(5-(6-Bromo-1H-indol-3-ylmethylene)-2-imino-1,3-dim...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250841(N-3'-ethylaplysinopsin | CHEMBL463250)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]methylspiperone form human cloned 5HT2A receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250840(5-(6-Bromo-1H-indol-3-ylmethylene)-2-imino-1,3-dim...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]methylspiperone form human cloned 5HT2A receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250839(CHEMBL2058413 | CHEMBL511879 | 6-bromo-2'-de-N-met...)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250841(N-3'-ethylaplysinopsin | CHEMBL463250)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50250839(CHEMBL2058413 | CHEMBL511879 | 6-bromo-2'-de-N-met...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]methylspiperone form human cloned 5HT2A receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed