Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50011970
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112776((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  93.1nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112782((1S,2R) Propane-2-sulfonic acid (2-phenyl-cyclopen...)
Affinity DataEC50:  551nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112772((R,R) Propane-2-sulfonic acid [2-(3,5-difluoro-phe...)
Affinity DataEC50:  281nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112770((R,R) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  22.6nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112780((+/-) Propane-2-sulfonic acid [2-(3-fluoro-phenyl)...)
Affinity DataEC50:  621nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112779((+/-) Propane-2-sulfonic acid [2-(4-nitro-phenyl)-...)
Affinity DataEC50:  190nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112781((R,R) Propane-2-sulfonic acid [2-(4-cyano-phenyl)-...)
Affinity DataEC50:  403nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112778((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  130nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112778((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  130nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112776((+/-) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  93.1nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112769((+/-) Propane-2-sulfonic acid [2-(3,4-difluoro-phe...)
Affinity DataEC50:  1.10E+3nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112775((+/-) Propane-2-sulfonic acid [2-(4-chloro-phenyl)...)
Affinity DataEC50:  247nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112777((+/-) Propane-2-sulfonic acid (2-p-tolyl-cyclopent...)
Affinity DataEC50:  434nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112773((+/-3b) N-{4'-[1-Methyl-2-(propane-2-sulfonylamino...)
Affinity DataEC50:  520nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112774((R,R) Propane-2-sulfonic acid (2-phenyl-cyclopenty...)
Affinity DataEC50:  1.74E+3nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112772((R,R) Propane-2-sulfonic acid [2-(3,5-difluoro-phe...)
Affinity DataEC50:  281nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112770((R,R) Propane-2-sulfonic acid [2-(4-iodo-phenyl)-c...)
Affinity DataEC50:  22.6nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50094024(propane-2-sulfonic acid [2-(4'-cyano-biphenyl-4-yl...)
Affinity DataEC50:  290nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed