Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50011990
TargetOxytocin receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(L-371257 | 1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-m...)
Affinity DataIC50: 640nMAssay Description:Compound was tested for displacement of 3[H] oxytocin from rat OT receptor (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50113051(N-{5-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperi...)
Affinity DataIC50: 744nMAssay Description:Compound was tested for displacement of 3[H] oxytocin from rat OT receptor (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50113050(N-{5-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperi...)
Affinity DataIC50: 3.04E+3nMAssay Description:Compound was tested for displacement of 3[H] oxytocin from rat OT receptor (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219760(CHEMBL286895)
Affinity DataKi:  0.501nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219779(CHEMBL30510)
Affinity DataKi:  1nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219786(CHEMBL285820)
Affinity DataKi:  1.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219762(CHEMBL283894)
Affinity DataKi:  2nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50113050(N-{5-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperi...)
Affinity DataKi:  2nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219774(CHEMBL281243)
Affinity DataKi:  2.5nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50113051(N-{5-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperi...)
Affinity DataKi:  3.20nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219775(CHEMBL31651)
Affinity DataKi:  3.20nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219776(CHEMBL32404)
Affinity DataKi:  4nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219509(CHEMBL287325)
Affinity DataKi:  6.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219764(CHEMBL281044)
Affinity DataKi:  6.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219783(CHEMBL282494)
Affinity DataKi:  6.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(L-371257 | 1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-m...)
Affinity DataKi:  6.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219785(CHEMBL283039)
Affinity DataKi:  6.30nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219781(CHEMBL30910)
Affinity DataKi:  7.90nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219761(CHEMBL287101)
Affinity DataKi:  7.90nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219770(CHEMBL283676)
Affinity DataKi:  10nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219782(CHEMBL281081)
Affinity DataKi:  10nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219773(CHEMBL445875)
Affinity DataKi:  10nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219780(CHEMBL287629)
Affinity DataKi:  25nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219777(CHEMBL281988)
Affinity DataKi:  25nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219771(CHEMBL281106)
Affinity DataKi:  50nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219769(CHEMBL286771)
Affinity DataKi:  63nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219784(CHEMBL282767)
Affinity DataKi:  79nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219778(CHEMBL287628)
Affinity DataKi:  100nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219765(CHEMBL30550)
Affinity DataKi:  100nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219787(CHEMBL30587)
Affinity DataKi:  794nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219768(CHEMBL31556)
Affinity DataKi:  794nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50113050(N-{5-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperi...)
Affinity DataKi:  1.26E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219762(CHEMBL283894)
Affinity DataKi:  1.59E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219774(CHEMBL281243)
Affinity DataKi:  1.59E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(L-371257 | 1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-m...)
Affinity DataKi: <2.00E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219772(CHEMBL29368)
Affinity DataKi: <3.16E+3nMAssay Description:Displacement of 3[H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50219776(CHEMBL32404)
Affinity DataKi:  3.98E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed