Compile Data Set for Download or QSAR
Report error Found 287 Enz. Inhib. hit(s) with all data for entry = 50003604
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataEC50:  0.110nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataEC50:  0.417nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  0.437nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  0.501nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataEC50:  0.912nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473682(CHEMBL70691)
Affinity DataEC50:  1.60nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataEC50:  1.90nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473671(CHEMBL71479)
Affinity DataEC50:  1.90nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataEC50:  2.20nMAssay Description:Agonist potency at alpha-1b adrenoceptors assayed in rat-1 fibroblasts expressing human alpha-1bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataEC50:  2.30nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  2.70nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  2.80nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473674(CHEMBL70634)
Affinity DataEC50:  2.80nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataEC50:  3.30nMAssay Description:Agonist potency at Alpha-2A stably expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473681(CHEMBL540035)
Affinity DataEC50:  3.40nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473682(CHEMBL70691)
Affinity DataEC50:  3.60nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataEC50:  4.60nMAssay Description:Agonist potency at Alpha-1A adrenoceptors assayed in rat-1 fibroblasts expressing human Alpha-1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataKi:  4.70nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataKi:  5nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473663(CHEMBL553276)
Affinity DataEC50:  5nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473682(CHEMBL70691)
Affinity DataEC50:  5nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataEC50:  5.60nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataEC50:  5.60nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473683(CHEMBL72724)
Affinity DataEC50:  6nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataEC50:  6nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataKi:  6.20nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  6.30nMAssay Description:Agonist potency at Alpha-2A stably expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataEC50:  7.80nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473669(CHEMBL70692)
Affinity DataEC50:  7.80nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473683(CHEMBL72724)
Affinity DataEC50:  7.90nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataEC50:  8.90nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor assayed in CHO cells expressing human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataEC50:  8.90nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataEC50:  9.10nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473683(CHEMBL72724)
Affinity DataEC50:  10nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataKi:  11nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473681(CHEMBL540035)
Affinity DataEC50:  14nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218568(CHEMBL71001)
Affinity DataEC50:  14nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataKi:  15nMAssay Description:Affinity to human Alpha-1B adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473669(CHEMBL70692)
Affinity DataEC50:  16nMAssay Description:Agonist potency at Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  16nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  16nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473684(CHEMBL74467)
Affinity DataEC50:  17nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataKi:  17nMAssay Description:Affinity to human Alpha-1D adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataKi:  18nMAssay Description:Affinity to human Alpha-2A adrenergic receptor determined by radioligand binding techniques from chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataKi:  19nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataEC50:  20nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataKi:  21nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataKi:  21nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataEC50:  22nMAssay Description:Agonist potency at Alpha-1D adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Glaxosmithkline Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473667(CHEMBL419448)
Affinity DataEC50:  24nMAssay Description:Agonist potency at Alpha-1 adrenergic receptor assayed in rat-1 fibroblasts expressing human Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
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