Compile Data Set for Download or QSAR
Report error Found 143 Enz. Inhib. hit(s) with all data for entry = 509
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 10nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 20nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 22nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 33nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 38nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 40nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 50nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3230(trans-4-[4-(2-Hydroxy-5,6,7,8-tetrahydro-1-naphtho...)
Affinity DataIC50: 50nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 50nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3235(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(trifluorome...)
Affinity DataIC50: 50nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 60nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 67nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3235(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(trifluorome...)
Affinity DataIC50: 100nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3236(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(methanesulf...)
Affinity DataIC50: 110nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3239(trans-2-[4-(6-Hydroxy-2-tetrazolylbenzoyl)-3,5-dih...)
Affinity DataIC50: 210nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3231((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 3,5...)
Affinity DataIC50: 250nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3239(trans-2-[4-(6-Hydroxy-2-tetrazolylbenzoyl)-3,5-dih...)
Affinity DataIC50: 260nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3230(trans-4-[4-(2-Hydroxy-5,6,7,8-tetrahydro-1-naphtho...)
Affinity DataIC50: 260nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3228(trans-4-[4-(2-Hydroxy-1-naphthoyl)-3,5-dihydroxybe...)
Affinity DataIC50: 290nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3220(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50: 290nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3230(trans-4-[4-(2-Hydroxy-5,6,7,8-tetrahydro-1-naphtho...)
Affinity DataIC50: 300nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3226(trans-4-[3,5-Dihydroxy-4-(4-hydroxy-3-phthlido)ben...)
Affinity DataIC50: 300nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3235(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(trifluorome...)
Affinity DataIC50: 310nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3220(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50: 320nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3234(2-(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxyben...)
Affinity DataIC50: 330nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3227(trans-3-(4-Hydroxybenzamido)-4-[3,5-dihydroxy-4-(2...)
Affinity DataIC50: 330nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3239(trans-2-[4-(6-Hydroxy-2-tetrazolylbenzoyl)-3,5-dih...)
Affinity DataIC50: 340nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3235(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(trifluorome...)
Affinity DataIC50: 350nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3216(trans-1-[4-(2-Carboxy-6-hydroxybenzoyl)-3-hydroxyb...)
Affinity DataIC50: 350nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3213((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 4-[...)
Affinity DataIC50: 360nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3220(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50: 370nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3234(2-(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxyben...)
Affinity DataIC50: 410nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3230(trans-4-[4-(2-Hydroxy-5,6,7,8-tetrahydro-1-naphtho...)
Affinity DataIC50: 430nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3211(4-trans-[4-(2-Hydroxybenzoyl)-3,5-dihydroxybenzoyl...)
Affinity DataIC50: 440nMpH: 7.5 T: 2°CAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3212((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 4-[...)
Affinity DataIC50: 440nMpH: 7.5 T: 2°CAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3220(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50: 460nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3241(trans-2-[4-[6-Hydroxy-2-(2-methyltetrazolyl)benzoy...)
Affinity DataIC50: 470nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3234(2-(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxyben...)
Affinity DataIC50: 470nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3225(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50: 470nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3232(trans-2-[4-(6-Hydroxy-2-nitrilobenzoyl)-3,5-dihydr...)
Affinity DataIC50: 500nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3236(trans-2-[3,5-Dihydroxy-4-[2-hydroxy-6-(methanesulf...)
Affinity DataIC50: 500nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3226(trans-4-[3,5-Dihydroxy-4-(4-hydroxy-3-phthlido)ben...)
Affinity DataIC50: 800nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Sphinx Laboratories

LigandPNGBDBM3232(trans-2-[4-(6-Hydroxy-2-nitrilobenzoyl)-3,5-dihydr...)
Affinity DataIC50: 830nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Sphinx Laboratories

LigandPNGBDBM3212((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 4-[...)
Affinity DataIC50: 860nMpH: 7.5 T: 2°CAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3207(CHEMBL193697 | 2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(...)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3215((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 1.20E+3nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Sphinx Laboratories

LigandPNGBDBM3240((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 1.30E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3217(3-hydroxy-2-{[4-({[(1R,2R)-2-[(4-hydroxybenzene)am...)
Affinity DataIC50: 1.70E+3nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
LigandPNGBDBM3240((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 1.80E+3nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2005
Entry Details Article
PubMed
Displayed 1 to 50 (of 143 total ) | Next | Last >>
Jump to: