Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012106
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114773(5-(Azetidin-2-ylmethoxy)-2-chloro-3-(2-pyridin-4-y...)
Affinity DataKi:  0.00900nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0100nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114771(2-Chloro-3-(2-pyridin-4-yl-ethyl)-5-(pyrrolidin-2-...)
Affinity DataKi:  0.0110nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114774(2-Chloro-3-(2-pyridin-4-yl-vinyl)-5-(pyrrolidin-2-...)
Affinity DataKi:  0.0150nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114768(2-Chloro-5-(1-methyl-pyrrolidin-2-ylmethoxy)-3-(2-...)
Affinity DataKi:  0.0230nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114767(2-Chloro-3-(2-pyridin-3-yl-vinyl)-5-(pyrrolidin-2-...)
Affinity DataKi:  0.0280nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114769(2-Chloro-5-(1-methyl-pyrrolidin-2-ylmethoxy)-3-(2-...)
Affinity DataKi:  0.0280nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114775(2-Chloro-5-(1-methyl-azetidin-2-ylmethoxy)-3-(2-py...)
Affinity DataKi:  0.0720nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114778(2-Chloro-5-(1-methyl-pyrrolidin-2-ylmethoxy)-3-(2-...)
Affinity DataKi:  0.0880nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114776(2-Chloro-5-(1-methyl-pyrrolidin-2-ylmethoxy)-3-(2-...)
Affinity DataKi:  0.265nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50114777(2-Chloro-3-(2-pyridin-2-yl-vinyl)-5-(pyrrolidin-2-...)
Affinity DataKi:  0.331nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed