Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50012125
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  8nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114973(N-(4-{[(Naphthalen-2-ylmethyl)-amino]-methyl}-cycl...)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50403914(CHEMBL2113711)
Affinity DataKi:  10nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114977(Naphthalene-1-sulfonic acid (4-{[(1,2,3,4-tetrahyd...)
Affinity DataKi:  11nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114979(Naphthalene-2-sulfonic acid (4-{[(1,2,3,4-tetrahyd...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114976(2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl...)
Affinity DataKi:  14nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114978(Naphthalene-1-sulfonic acid (4-{[2-(4-chloro-pheny...)
Affinity DataKi:  17nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  18nMAssay Description:Functional response of NPY to inhibit forskolin-stimulated cAMP in cells stably transfected with rat Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114981(N-(4-{[(Naphthalen-1-ylmethyl)-amino]-methyl}-cycl...)
Affinity DataKi:  26nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114980(2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl...)
Affinity DataKi:  28nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  63nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  100nMAssay Description:Bnding affinity against cloned human Alpha-2C adrenergic receptor was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114975(Naphthalene-2-sulfonic acid {6-[(naphthalen-2-ylme...)
Affinity DataKi:  123nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114978(Naphthalene-1-sulfonic acid (4-{[2-(4-chloro-pheny...)
Affinity DataKi:  3.24E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114977(Naphthalene-1-sulfonic acid (4-{[(1,2,3,4-tetrahyd...)
Affinity DataKi:  3.55E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114979(Naphthalene-2-sulfonic acid (4-{[(1,2,3,4-tetrahyd...)
Affinity DataKi:  5.55E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114975(Naphthalene-2-sulfonic acid {6-[(naphthalen-2-ylme...)
Affinity DataKi:  7.30E+3nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114973(N-(4-{[(Naphthalen-2-ylmethyl)-amino]-methyl}-cycl...)
Affinity DataKi:  1.30E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114981(N-(4-{[(Naphthalen-1-ylmethyl)-amino]-methyl}-cycl...)
Affinity DataKi:  1.45E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  1.60E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50403914(CHEMBL2113711)
Affinity DataKi:  1.72E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Rat)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114974(2-nitro-N-((4-(((1,2,3,4-tetrahydronaphthalen-2-yl...)
Affinity DataKi:  2.20E+4nMAssay Description:Functional response of NPY to inhibit forskolin-stimulated cAMP in cells stably transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114976(2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl...)
Affinity DataKi:  2.37E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50114980(2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl...)
Affinity DataKi:  4.87E+4nMAssay Description:Tested for radioligand binding affinity against membranes from COS-7 cells transiently transfected with Neuropeptide Y receptor type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed