Compile Data Set for Download or QSAR
Report error Found 183 Enz. Inhib. hit(s) with all data for entry = 50012192
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14157(N-(4-carbamimidoylphenyl)-2-hydroxy-3-iodo-5-methy...)
Affinity DataKi:  80nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115894(3-Hydroxy-anthracene-2-carboxylic acid (6-guanidin...)
Affinity DataKi:  85nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14156(CHEMBL61327 | 3-bromo-N-(4-carbamimidoylphenyl)-2-...)
Affinity DataKi:  150nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115896(3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic aci...)
Affinity DataKi:  180nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115907(3-Hydroxy-anthracene-2-carboxylic acid (4-carbamim...)
Affinity DataKi:  190nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50098137(CHEMBL60088 | 2-amidino-4-iodobenzothiophene | CHE...)
Affinity DataKi:  210nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115889(4-Bromo-3-hydroxy-anthracene-2-carboxylic acid (6-...)
Affinity DataKi:  220nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115902(3-Hydroxy-4-isopropoxy-anthracene-2-carboxylic aci...)
Affinity DataKi:  230nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14157(N-(4-carbamimidoylphenyl)-2-hydroxy-3-iodo-5-methy...)
Affinity DataKi:  240nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115898(3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (...)
Affinity DataKi:  250nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14158(CHEMBL293260 | N-(4-carbamimidoyl-3-fluorophenyl)-...)
Affinity DataKi:  270nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14156(CHEMBL61327 | 3-bromo-N-(4-carbamimidoylphenyl)-2-...)
Affinity DataKi:  280nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115905(3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (...)
Affinity DataKi:  280nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14157(N-(4-carbamimidoylphenyl)-2-hydroxy-3-iodo-5-methy...)
Affinity DataKi:  290nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115891(3-Hydroxy-anthracene-2-carboxylic acid (4-guanidin...)
Affinity DataKi:  300nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14156(CHEMBL61327 | 3-bromo-N-(4-carbamimidoylphenyl)-2-...)
Affinity DataKi:  360nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14157(N-(4-carbamimidoylphenyl)-2-hydroxy-3-iodo-5-methy...)
Affinity DataKi:  380nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14158(CHEMBL293260 | N-(4-carbamimidoyl-3-fluorophenyl)-...)
Affinity DataKi:  410nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14156(CHEMBL61327 | 3-bromo-N-(4-carbamimidoylphenyl)-2-...)
Affinity DataKi:  440nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14157(N-(4-carbamimidoylphenyl)-2-hydroxy-3-iodo-5-methy...)
Affinity DataKi:  460nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14158(CHEMBL293260 | N-(4-carbamimidoyl-3-fluorophenyl)-...)
Affinity DataKi:  520nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115895(N-(4-Carbamimidoyl-phenyl)-3-chloro-2-hydroxy-benz...)
Affinity DataKi:  600nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115903(N-(4-Carbamimidoyl-phenyl)-4-ethoxy-2-hydroxy-benz...)
Affinity DataKi:  650nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115899(3-Hydroxy-4-iodo-anthracene-2-carboxylic acid (6-g...)
Affinity DataKi:  700nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115886(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-4-methyl-benz...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115895(N-(4-Carbamimidoyl-phenyl)-3-chloro-2-hydroxy-benz...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115895(N-(4-Carbamimidoyl-phenyl)-3-chloro-2-hydroxy-benz...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115895(N-(4-Carbamimidoyl-phenyl)-3-chloro-2-hydroxy-benz...)
Affinity DataKi:  1.50E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115880(4-Bromo-3-hydroxy-anthracene-2-carboxylic acid (4-...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115908(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-3-methyl-benz...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14158(CHEMBL293260 | N-(4-carbamimidoyl-3-fluorophenyl)-...)
Affinity DataKi:  1.70E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115907(3-Hydroxy-anthracene-2-carboxylic acid (4-carbamim...)
Affinity DataKi:  1.80E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115903(N-(4-Carbamimidoyl-phenyl)-4-ethoxy-2-hydroxy-benz...)
Affinity DataKi:  2.00E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115886(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-4-methyl-benz...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50102768(2-(2-Hydroxy-phenyl)-1H-indole-5-carboxamidine | C...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115901(N-(4-Carbamimidoyl-phenyl)-4-chloro-2-hydroxy-benz...)
Affinity DataKi:  2.40E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115878(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-5-methyl-benz...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14155(N-(4-CARBAMIMIDOYL-PHENYL)-2-HYDROXY-BENZAMIDE | N...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115901(N-(4-Carbamimidoyl-phenyl)-4-chloro-2-hydroxy-benz...)
Affinity DataKi:  2.80E+3nMAssay Description:The compound was evaluated to inhibit the Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115910(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-5-methoxy-ben...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115886(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-4-methyl-benz...)
Affinity DataKi:  3.60E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115908(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-3-methyl-benz...)
Affinity DataKi:  3.90E+3nMAssay Description:Activation of plasminogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115907(3-Hydroxy-anthracene-2-carboxylic acid (4-carbamim...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14156(CHEMBL61327 | 3-bromo-N-(4-carbamimidoylphenyl)-2-...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115877(3-Hydroxy-4-iodo-anthracene-2-carboxylic acid (4-g...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115910(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-5-methoxy-ben...)
Affinity DataKi:  5.20E+3nMAssay Description:The compound was evaluated to inhibit the Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM14158(CHEMBL293260 | N-(4-carbamimidoyl-3-fluorophenyl)-...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50100897(2-{5-[AMINO(IMINIO)METHYL]-1H-BENZIMIDAZOL-2-YL}BE...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115884(N-(4-Guanidino-phenyl)-2-hydroxy-4-methyl-benzamid...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Celera

Curated by ChEMBL
LigandPNGBDBM50115908(N-(4-Carbamimidoyl-phenyl)-2-hydroxy-3-methyl-benz...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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