Compile Data Set for Download or QSAR
Report error Found 117 Enz. Inhib. hit(s) with all data for entry = 50037063
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118272(5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidaz...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 1nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055017(7,8-Dichloro-5-(4-chloro-phenyl)-2,5-dihydro-3H-im...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataIC50: 1.09nMAssay Description:Inhibition of [3H]WIN-35428 radioligand binding to the Dopamine Transporter in guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118263(5-(4-Chloro-phenyl)-7-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 1.46nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataKi:  1.70nMAssay Description:Ability to displace [125I]- RTI-55 binding at the Dopamine transporter site on HEK cells expressing cDNA for the human transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118268(5-(4-Chloro-phenyl)-6-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 1.73nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118260(9-(4-Hydroxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataIC50: 1.94nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataIC50: 2.21nMAssay Description:Ability to block the uptake of 5-HT at the Dopamine transporter of HEK cells expressing cDNA for the human transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118262(9-(4-Methoxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataIC50: 2.5nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataKi:  2.55nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055019(5-Phenyl-2,5-dihydro-3H-imidazo[2,1-a]isoindol-5-o...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118265(5-(4-Chloro-phenyl)-9-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118260(9-(4-Hydroxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataIC50: 3.40nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118262(9-(4-Methoxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 4.20nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter in guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118265(5-(4-Chloro-phenyl)-9-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118265(5-(4-Chloro-phenyl)-9-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 4.75nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine Transporter of guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50005536(Mazanor | 42-548 | 5-(4-Chloro-phenyl)-2,5-dihydro...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118272(5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidaz...)
Affinity DataIC50: 5nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118263(5-(4-Chloro-phenyl)-7-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055017(7,8-Dichloro-5-(4-chloro-phenyl)-2,5-dihydro-3H-im...)
Affinity DataIC50: 6nMAssay Description:Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataIC50: 6nMAssay Description:Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118265(5-(4-Chloro-phenyl)-9-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50005536(Mazanor | 42-548 | 5-(4-Chloro-phenyl)-2,5-dihydro...)
Affinity DataIC50: 8.10nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataKi:  8.80nMAssay Description:Ability to displace [125I]- RTI-55 binding at the Norepinephrine transporter site on HEK cells expressing cDNA for the human transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055017(7,8-Dichloro-5-(4-chloro-phenyl)-2,5-dihydro-3H-im...)
Affinity DataIC50: 10nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118268(5-(4-Chloro-phenyl)-6-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  10.3nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118272(5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidaz...)
Affinity DataIC50: 12.3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine Transporter of guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118263(5-(4-Chloro-phenyl)-7-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 13.3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine Transporter of guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055017(7,8-Dichloro-5-(4-chloro-phenyl)-2,5-dihydro-3H-im...)
Affinity DataIC50: 13.6nMAssay Description:Ability to displace [3H]WIN-35428 from Dopamine Transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataIC50: 15nMAssay Description:Inhibition of 5-HT uptake in HEK cells expressing human serotonin transporter (hSERT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118263(5-(4-Chloro-phenyl)-7-methoxy-2,5-dihydro-3H-imida...)
Affinity DataIC50: 16.7nMAssay Description:Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50005536(Mazanor | 42-548 | 5-(4-Chloro-phenyl)-2,5-dihydro...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055003(9-(4-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118263(5-(4-Chloro-phenyl)-7-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118268(5-(4-Chloro-phenyl)-6-methoxy-2,5-dihydro-3H-imida...)
Affinity DataKi:  23.1nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118272(5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidaz...)
Affinity DataKi:  23.1nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118266(9-Benzo[1,3]dioxol-5-yl-1,2,3,9-tetrahydro-4,9a-di...)
Affinity DataKi:  25.6nMAssay Description:Displacement of [125I]- RTI-55 from Serotonin transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]- RTI-55 from Serotonin transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118269(5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]i...)
Affinity DataIC50: 29.7nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine Transporter of guinea pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118262(9-(4-Methoxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataIC50: 30.4nMAssay Description:Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118262(9-(4-Methoxy-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza...)
Affinity DataKi:  36.2nMAssay Description:Displacement of [125I]- RTI-55 from Dopamine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Drew University

Curated by ChEMBL
LigandPNGBDBM50118272(5-(4-Chloro-phenyl)-9-fluoro-2,5-dihydro-3H-imidaz...)
Affinity DataKi:  38.1nMAssay Description:Displacement of [125I]- RTI-55 from Serotonin transporter expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
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