Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50041324
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | Chlorochin | CHLOROQUINE PHOSPHATE | Chlo...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120736((2-Piperidin-1-yl-ethyl)-(7-trifluoromethyl-quinol...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120735(N1-tert-butyl-N2-(7-chloroquinolin-4-yl)ethane-1,2...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120737(N-tert-Butyl-N'-(7-trifluoromethyl-quinolin-4-yl)-...)
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120738(7-chloro-N-(2-(pyrrolidin-1-yl)ethyl)quinolin-4-am...)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120734((7-Chloro-quinolin-4-yl)-(2-piperidin-1-yl-ethyl)-...)
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetHistidine-rich protein PFHRP-II(malaria parasite P. falciparum)
The University of Liverpool

Curated by ChEMBL
LigandPNGBDBM50120739((7-Chloro-quinolin-4-yl)-(2-morpholin-4-yl-ethyl)-...)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of beta-hematin formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed