Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50012614
TargetProcathepsin L(Rat)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121030([(S)-1-((5S,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 4nMAssay Description:In vitro Inhibitory activity against Cathepsin L cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121030([(S)-1-((5S,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 5nMAssay Description:In vitro Inhibitory activity against Cathepsin K cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121030([(S)-1-((5S,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 77nMAssay Description:In vitro Inhibitory activity against Cathepsin S cysteine protease by using Cbz-Val-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Rat)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121028([(S)-1-((S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept-6...)
Affinity DataIC50: 85nMAssay Description:In vitro Inhibitory activity against Cathepsin L cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121031([(S)-2-Methyl-1-((5R,6S)-7-oxo-4-oxa-1-aza-bicyclo...)
Affinity DataIC50: 100nMAssay Description:In vitro Inhibitory activity against Cathepsin K cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121031([(S)-2-Methyl-1-((5R,6S)-7-oxo-4-oxa-1-aza-bicyclo...)
Affinity DataIC50: 260nMAssay Description:In vitro Inhibitory activity against Cathepsin S cysteine protease by using Cbz-Val-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121028([(S)-1-((S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept-6...)
Affinity DataIC50: 430nMAssay Description:In vitro Inhibitory activity against Cathepsin S cysteine protease by using Cbz-Val-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Rat)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121031([(S)-2-Methyl-1-((5R,6S)-7-oxo-4-oxa-1-aza-bicyclo...)
Affinity DataIC50: 600nMAssay Description:In vitro Inhibitory activity against Cathepsin L cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121028([(S)-1-((S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept-6...)
Affinity DataIC50: 1.63E+3nMAssay Description:In vitro Inhibitory activity against Cathepsin K cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121028([(S)-1-((S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept-6...)
Affinity DataIC50: 1.76E+3nMAssay Description:In vitro Inhibitory activity against Cathepsin B cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Rat)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121029([(S)-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept...)
Affinity DataIC50: 1.83E+3nMAssay Description:In vitro Inhibitory activity against Cathepsin L cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121032([(S)-1-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro Inhibitory activity against Cathepsin S cysteine protease by using Cbz-Val-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121032([(S)-1-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro Inhibitory activity against Cathepsin K cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121030([(S)-1-((5S,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 1.22E+4nMAssay Description:In vitro Inhibitory activity against Cathepsin B cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121031([(S)-2-Methyl-1-((5R,6S)-7-oxo-4-oxa-1-aza-bicyclo...)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro Inhibitory activity against Cathepsin B cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Rat)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121032([(S)-1-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 3.80E+4nMAssay Description:In vitro Inhibitory activity against Cathepsin L cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121029([(S)-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]hept...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro Inhibitory activity against Cathepsin B cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Currently Naeja Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121032([(S)-1-((5R,6S)-7-Oxo-4-oxa-1-aza-bicyclo[3.2.0]he...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro Inhibitory activity against Cathepsin B cysteine protease by using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed