Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50012755
Affinity DataKd: 2nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataKd: 8nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 8nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 8nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Transcriptional activation assay in CV-1 cells expressing human retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]ATRA binding to human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Agonistic activity against Retinoic acid receptor RAR beta in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Inhibition of [3H]ATRA binding to human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Inhibition of [3H]9-cis-RA binding to mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 22nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 53nMAssay Description:Inhibition of [3H]9-cis-RA binding to human Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 78nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 93nMAssay Description:Inhibition of [3H]ATRA binding to human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Inhibition of [3H]-ATRA binding to human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 124nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 128nMAssay Description:Transcriptional activation in CV-1 cells expressing mouse Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 139nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 148nMAssay Description:Inhibition of [3H]ATRA binding to human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 153nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair





3D Structure (crystal)
