Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50035365
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | Tyr-Pro-Phe-Pro-NH2 | [D-Pro4]morph...)
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125255((R)-2-[((S)-1-{(R)-6-Amino-2-[(S)-2-({(S)-1-[(S)-2...)
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125259(Neuropeptide Y[24-36] | CHEMBL410260)
Affinity DataIC50: 6.90E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibitory activity against non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125256(Neuropeptide Y[22-36] | CHEMBL428276)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125258((S)-1-[(S)-6-Amino-2-((S)-2-{[(S)-1-((S)-2-amino-3...)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | Tyr-Pro-Phe-Pro-NH2 | [D-Pro4]morph...)
Affinity DataKi:  150nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125255((R)-2-[((S)-1-{(R)-6-Amino-2-[(S)-2-({(S)-1-[(S)-2...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125259(Neuropeptide Y[24-36] | CHEMBL410260)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  4.80E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125256(Neuropeptide Y[22-36] | CHEMBL428276)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of North Carolina At Wilmington

Curated by ChEMBL
LigandPNGBDBM50125258((S)-1-[(S)-6-Amino-2-((S)-2-{[(S)-1-((S)-2-amino-3...)
Affinity DataKi:  7.50E+3nMAssay Description:Binding affinity towards non-selective opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2012
Entry Details Article
PubMed