Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50013036
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125738(8a-Benzyloxymethyl-2-(2-cyclohex-1-enyl-ethyl)-6-f...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125738(8a-Benzyloxymethyl-2-(2-cyclohex-1-enyl-ethyl)-6-f...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125740(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125741(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125740(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125741(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125736(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 760nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125736(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 770nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125735(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125735(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125733(6-Furan-2-yl-8a-hydroxymethyl-1,4-dioxo-2-(4-pheny...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125739(2-Allyl-8a-benzyloxymethyl-6-furan-2-yl-1,4-dioxo-...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125733(6-Furan-2-yl-8a-hydroxymethyl-1,4-dioxo-2-(4-pheny...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibitory activity against Human Hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by HSL [14 C] cholesteryl oleate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125739(2-Allyl-8a-benzyloxymethyl-6-furan-2-yl-1,4-dioxo-...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125734(8a-Benzyloxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-phe...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125742(8a-tert-Butoxymethyl-6-furan-2-yl-1,4-dioxo-2-(4-p...)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHormone-sensitive lipase(Human)
Ontogen

Curated by ChEMBL
LigandPNGBDBM50125737(8a-Benzyloxymethyl-2-(2-cyclohex-1-enyl-ethyl)-6-f...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against human hormone-sensitive lipase (HSL) expressed in the baculovirus was determined by p-nitrophenyl butyrate (PNPB) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed