Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50013083
LigandPNGBDBM50126336(4-{[(4-Cyano-3-naphthalen-1-yl-phenyl)-(3-methyl-3...)
Affinity DataIC50: 0.370nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126339(4-[(3-CYANO-BENZYL)-(3-METHYL-3H-IMIDAZOL-4-YLMETH...)
Affinity DataIC50: 0.390nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50126340(4-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 0.450nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126335(R-115777 | 6-[(S)-AMINO(4-CHLOROPHENYL)(1-METHYL-1...)
Affinity DataIC50: 0.570nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126330(5-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 0.970nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM17325(CHEMBL29982 | (2S)-2-[(4-{[butyl(2-cyclohexylethyl...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126337(4-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126331(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126331(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126333(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50: 1.90nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)
Affinity DataIC50: 7.80nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126334(5-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126344(5-[Benzyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126329(N-(4-Cyano-3-naphthalen-1-yl-phenyl)-N-(3-methyl-3...)
Affinity DataIC50: 14nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126338(N-(4-Cyano-3-naphthalen-1-yl-phenyl)-N-(3-methyl-3...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126328(4-[(3-Methyl-3H-imidazol-4-ylmethyl)-amino]-2-naph...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126328(4-[(3-Methyl-3H-imidazol-4-ylmethyl)-amino]-2-naph...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126341(4-[Methyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126341(4-[Methyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126343(5-[Benzyloxy-(3-methyl-3H-imidazol-4-yl)-methyl]-2...)
Affinity DataIC50: 65nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126332(5-[Benzyl-(3H-imidazol-4-ylmethyl)-amino]-2'-methy...)
Affinity DataIC50: 84nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126339(4-[(3-CYANO-BENZYL)-(3-METHYL-3H-IMIDAZOL-4-YLMETH...)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50126333(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126340(4-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126329(N-(4-Cyano-3-naphthalen-1-yl-phenyl)-N-(3-methyl-3...)
Affinity DataIC50: 310nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126336(4-{[(4-Cyano-3-naphthalen-1-yl-phenyl)-(3-methyl-3...)
Affinity DataIC50: 650nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126334(5-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126337(4-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126342(2'-Methyl-5-[(3-methyl-3H-imidazol-4-ylmethyl)-ami...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126330(5-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126338(N-(4-Cyano-3-naphthalen-1-yl-phenyl)-N-(3-methyl-3...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed