Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50013122
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  0.700nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126814(1-(4-(trifluoromethyl)benzyl)-4-(2-(bis(4-fluoroph...)
Affinity DataKi:  1.10nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126823(1-(4-bromobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  1.10nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126813(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-c...)
Affinity DataKi:  1.20nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126820(1-(4-nitrobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  1.20nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126817(4-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperid...)
Affinity DataKi:  1.20nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126815(1-(4-iodobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy)...)
Affinity DataKi:  2.10nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126822(1-(4-fluorobenzyl)-4-(2-(bis(4-fluorophenyl)methox...)
Affinity DataKi:  2.30nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055882(4-(2-Benzhydryloxy-ethyl)-1-(4-nitro-benzyl)-piper...)
Affinity DataKi:  2.5nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055882(4-(2-Benzhydryloxy-ethyl)-1-(4-nitro-benzyl)-piper...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098405(4-(2-Benzhydryloxy-ethyl)-1-(4-trifluoromethyl-ben...)
Affinity DataKi:  3.5nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  3.70nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50126822(1-(4-fluorobenzyl)-4-(2-(bis(4-fluorophenyl)methox...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055879(4-(2-Benzhydryloxy-ethyl)-1-(4-chloro-benzyl)-pipe...)
Affinity DataKi:  3.80nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055876(4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benzyl)-pipe...)
Affinity DataKi:  5.10nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055871(4-(2-Benzhydryloxy-ethyl)-1-(4-bromo-benzyl)-piper...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50098393(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataKi:  5.70nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126816(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-m...)
Affinity DataKi:  5.70nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50055871(4-(2-Benzhydryloxy-ethyl)-1-(4-bromo-benzyl)-piper...)
Affinity DataKi:  6.40nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126820(1-(4-nitrobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  6.90nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)
Affinity DataKi:  7.20nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126819(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-m...)
Affinity DataKi:  7.90nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049365(1-benzyl-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pi...)
Affinity DataKi:  9.90nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126818(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-m...)
Affinity DataKi:  13.3nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126815(1-(4-iodobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy)...)
Affinity DataKi:  13.6nMAssay Description:Inhibition of [3H]dopamine uptake via rat dopamine receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50118602(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-naph...)
Affinity DataKi:  16nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126821(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(2-m...)
Affinity DataKi:  63nMAssay Description:Affinity at rat dopamine transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  73nMAssay Description:Inhibition of [3H]5-HT uptake at the rat serotonin transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  79nMAssay Description:Inhibition of [3H]norepinephrine uptake at the rat norepinephrine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  88nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  93nMAssay Description:Inhibition of [3H]norepinephrine uptake at the rat norepinephrine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  126nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126818(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(3-m...)
Affinity DataKi:  161nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50049365(1-benzyl-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pi...)
Affinity DataKi:  171nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126823(1-(4-bromobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  199nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126815(1-(4-iodobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy)...)
Affinity DataKi:  205nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055882(4-(2-Benzhydryloxy-ethyl)-1-(4-nitro-benzyl)-piper...)
Affinity DataKi:  208nMAssay Description:Inhibition of [3H]norepinephrine uptake at the rat norepinephrine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  227nMAssay Description:Inhibition of [3H]5-HT uptake at the rat serotonin transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Niddk

Curated by ChEMBL
LigandPNGBDBM50126820(1-(4-nitrobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  231nMAssay Description:Inhibition of [3H]norepinephrine uptake at the rat norepinephrine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126813(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-c...)
Affinity DataKi:  238nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126816(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-m...)
Affinity DataKi:  239nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126822(1-(4-fluorobenzyl)-4-(2-(bis(4-fluorophenyl)methox...)
Affinity DataKi:  245nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126821(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(2-m...)
Affinity DataKi:  248nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126819(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-m...)
Affinity DataKi:  266nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50118602(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-naph...)
Affinity DataKi:  370nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126820(1-(4-nitrobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  387nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50126814(1-(4-(trifluoromethyl)benzyl)-4-(2-(bis(4-fluoroph...)
Affinity DataKi:  442nMAssay Description:Affinity at rat serotonin transporter using [125I]RTI-55 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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