Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50037248
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126888(CHEMBL193978 | CHEMBL416053 | 1-[4-(4-Piperidin-1-...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126878(1-[4-(4-Imidazol-1-yl-phenoxymethyl)-benzyl]-piper...)
Affinity DataKd:  15.8nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126902(1-[4-(4-Pyrrolidin-1-ylmethyl-benzyloxy)-phenyl]-e...)
Affinity DataKd:  18.2nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126902(1-[4-(4-Pyrrolidin-1-ylmethyl-benzyloxy)-phenyl]-e...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126878(1-[4-(4-Imidazol-1-yl-phenoxymethyl)-benzyl]-piper...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126875(Cyclopentyl-[4-(4-piperidin-1-ylmethyl-benzyloxy)-...)
Affinity DataKd:  30.9nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126900(1-[4-(4-Azepan-1-ylmethyl-benzyloxy)-phenyl]-ethan...)
Affinity DataKd:  30.9nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126900(1-[4-(4-Azepan-1-ylmethyl-benzyloxy)-phenyl]-ethan...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126888(CHEMBL193978 | CHEMBL416053 | 1-[4-(4-Piperidin-1-...)
Affinity DataKd:  38.0nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50089295(1-[5-(4-Nitro-phenoxy)-pentyl]-pyrrolidine | 1-[5-...)
Affinity DataKi:  39nMAssay Description:In vivo binding affinity was determined by measuring the displacement curves of [125I]iodoproxyfan in human Histamine H3 receptor antagonist with rel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126903(1-[4-(4-Chloro-3-methyl-phenoxymethyl)-benzyl]-pip...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  46nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126895(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126884(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  61.7nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126886(Cyclopropyl-[4-(4-piperidin-1-ylmethyl-benzyloxy)-...)
Affinity DataKi:  66nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126884(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKi:  84nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126895(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  85.1nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126890(1-[4-(Indan-5-yloxymethyl)-benzyl]-piperidine; com...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126883(1-{4-[3-(1H-Imidazol-4-yl)-propoxymethyl]-phenyl}-...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126905(1-[4-(4-Propoxy-phenoxymethyl)-benzyl]-piperidine;...)
Affinity DataKi:  88nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126898(Phenyl-[4-(4-piperidin-1-ylmethyl-benzyloxy)-benzy...)
Affinity DataKi:  90nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126879(1-[4-(4-Diethylaminomethyl-benzyloxy)-phenyl]-etha...)
Affinity DataKi:  91nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126881(1-[4-(5,6,7,8-Tetrahydro-naphthalen-2-yloxymethyl)...)
Affinity DataKi:  92nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126891(1-[4-(4-Chloro-3-fluoro-phenoxymethyl)-benzyl]-pip...)
Affinity DataKi:  95nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126882(1-[4-(4-Iodo-phenoxymethyl)-benzyl]-piperidine; co...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126893(1-[4-(4-Bromo-phenoxymethyl)-benzyl]-piperidine; c...)
Affinity DataKi:  114nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126901(1-[4-(4-Methoxy-phenoxymethyl)-benzyl]-piperidine;...)
Affinity DataKi:  119nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126885(1-[4-(4-Fluoro-phenoxymethyl)-benzyl]-piperidine; ...)
Affinity DataKi:  123nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126887(1-[4-(4-Chloro-phenoxymethyl)-benzyl]-piperidine; ...)
Affinity DataKi:  124nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126911(1-[4-(4-Trifluoromethyl-phenoxymethyl)-benzyl]-pip...)
Affinity DataKi:  125nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126909(1-(4-p-Tolyloxymethyl-benzyl)-piperidine; compound...)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126899(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKi:  129nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126910(1-[4-(3,4-Dimethyl-phenoxymethyl)-benzyl]-piperidi...)
Affinity DataKi:  149nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126875(Cyclopentyl-[4-(4-piperidin-1-ylmethyl-benzyloxy)-...)
Affinity DataKi:  157nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126904(1-[4-(4-Ethyl-phenoxymethyl)-benzyl]-piperidine; c...)
Affinity DataKi:  163nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126906(1-[4-(3,4-Dichloro-phenoxymethyl)-benzyl]-piperidi...)
Affinity DataKi:  167nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126907(1-[4-(4-Butyl-phenoxymethyl)-benzyl]-piperidine; c...)
Affinity DataKi:  169nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126873(1-[4-(4-Cyclopentyl-phenoxymethyl)-benzyl]-piperid...)
Affinity DataKi:  201nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126889(1-(4-Phenoxymethyl-benzyl)-piperidine; compound wi...)
Affinity DataKi:  227nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126876(1-[4-(4-Benzyl-phenoxymethyl)-benzyl]-piperidine; ...)
Affinity DataKi:  238nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126880(1-[4-(4-Isopropyl-phenoxymethyl)-benzyl]-piperidin...)
Affinity DataKi:  253nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126908(1-[4-(4-Propyl-phenoxymethyl)-benzyl]-piperidine; ...)
Affinity DataKi:  257nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126899(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  288nMAssay Description:Potency at histamine H3 receptor subtype, was tested on guinea pig right ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126896(1-(4-m-Tolyloxymethyl-benzyl)-piperidine; compound...)
Affinity DataKi:  334nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126894(1-[4-(4-Phenoxy-phenoxymethyl)-benzyl]-piperidine;...)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126897(1-[4-(4-Benzyloxy-phenoxymethyl)-benzyl]-piperidin...)
Affinity DataKi:  550nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126874(1-[4-(4-Styryl-phenoxymethyl)-benzyl]-piperidine; ...)
Affinity DataKi:  761nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50126877(1-[4-(4-Phenethyl-phenoxymethyl)-benzyl]-piperidin...)
Affinity DataKi:  890nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
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