Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 5242
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85592(AANAT Inhibitor, 12d)
Affinity DataIC50: 180nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85590(AANAT Inhibitor, 8h)
Affinity DataIC50: 390nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85587(AANAT Inhibitor, 8d)
Affinity DataIC50: 610nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85588(AANAT Inhibitor, 8e)
Affinity DataIC50: 680nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85591(AANAT Inhibitor, 8i)
Affinity DataIC50: 700nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM50282747(CHEMBL290406 | AANAT Inhibitor, 1 | 2-Bromo-N-[2-(...)
Affinity DataIC50: 1.43E+3nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85589(AANAT Inhibitor, 8g)
Affinity DataIC50: 3.78E+3nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSerotonin N-acetyltransferase(Human)
UniversitÉ

LigandPNGBDBM85586(AANAT Inhibitor, 8c)
Affinity DataIC50: 4.00E+4nMpH: 6.8 T: 2°CAssay Description:The compounds were evaluated in a human serotonin N-acetyltransferase assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed