Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50013221
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127832(3-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50120543(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127844(3-Ethyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-in...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50120542(2-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-imidazo[1,...)
Affinity DataKi:  6nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127831(2-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-pyrazolo[1...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127838(1-Methyl-2-[2-methyl-4-(3-piperidin-1-yl-propoxy)-...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127841(2-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-indolizine...)
Affinity DataKi:  13nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127834(1-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  16nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127839(1-Methanesulfonyl-2-[4-(3-piperidin-1-yl-propoxy)-...)
Affinity DataKi:  16nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127840(1-Ethyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-in...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127830(6-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  28nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127835(1-Phenethyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl...)
Affinity DataKi:  37nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127846(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127847(1-Phenyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127833(8-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127843(5-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  46nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127837(2-[4-(3-Piperidin-1-yl-propoxy)-phenyl]-1H-indole ...)
Affinity DataKi:  47nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127845(2-[2-Methyl-4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  152nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127836(2-[2-(3-Piperidin-1-yl-propoxy)-phenyl]-indolizine...)
Affinity DataKi:  236nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50127842(2-[3-(3-Piperidin-1-yl-propoxy)-phenyl]-indolizine...)
Affinity DataKi:  308nMAssay Description:Binding affinity towards human Histamine H3 receptor using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed