Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 915
LigandPNGBDBM7240((3Z)-N-methyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7244((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7254((3Z)-N-methyl-2-oxo-3-({4-oxo-2H,4H,5H,6H,7H-pyrro...)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7250((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7241((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7249((3Z)-4-(2-hydroxyethyl)-3-({4-oxo-2H,4H,6H,7H-pyra...)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7243((3Z)-N,N-dimethyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyra...)
Affinity DataIC50: 33nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7239((3Z)-5-methoxy-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7260((3Z)-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,4-c]pyridi...)
Affinity DataIC50: 49nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7242((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 64nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7256((3Z)-2-oxo-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,4-c]...)
Affinity DataIC50: 68nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7255((3Z)-N,N-dimethyl-2-oxo-3-({4-oxo-2H,4H,5H,6H,7H-p...)
Affinity DataIC50: 68nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7245((3Z)-5-fluoro-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 82nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7246((3Z)-5-chloro-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 88nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataIC50: 110nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataIC50: 130nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7247((3Z)-5-bromo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]py...)
Affinity DataIC50: 190nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7253((3Z)-5-methoxy-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,...)
Affinity DataIC50: 250nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7248((3Z)-4-methyl-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 270nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7257((3Z)-5-fluoro-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,4...)
Affinity DataIC50: 300nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7259((3Z)-4-(2-hydroxyethyl)-3-({4-oxo-2H,4H,5H,6H,7H-p...)
Affinity DataIC50: 340nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7250((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 490nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7258((3Z)-5-bromo-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,4-...)
Affinity DataIC50: 530nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7250((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 1.10E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7252((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 1.10E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7250((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 1.10E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7249((3Z)-4-(2-hydroxyethyl)-3-({4-oxo-2H,4H,6H,7H-pyra...)
Affinity DataIC50: 1.20E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7251((3Z)-6-methoxy-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]...)
Affinity DataIC50: 1.40E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7251((3Z)-6-methoxy-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]...)
Affinity DataIC50: 1.50E+3nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7252((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 2.00E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7246((3Z)-5-chloro-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 2.10E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7261((3Z)-3-({4-oxo-2H,4H,5H,6H,7H-pyrrolo[3,4-c]pyridi...)
Affinity DataIC50: 5.70E+3nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7244((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 6.20E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7240((3Z)-N-methyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3...)
Affinity DataIC50: 6.60E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7241((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 6.60E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7242((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 6.70E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7252((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 8.40E+3nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7252((3Z)-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrrol-1-y...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7245((3Z)-5-fluoro-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataIC50: 1.10E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7247((3Z)-5-bromo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]py...)
Affinity DataIC50: 1.10E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7241((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 1.30E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataIC50: 1.80E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7247((3Z)-5-bromo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]py...)
Affinity DataIC50: 1.80E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7240((3Z)-N-methyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7243((3Z)-N,N-dimethyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyra...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7242((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7243((3Z)-N,N-dimethyl-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyra...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7244((3Z)-2-oxo-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]pyrr...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
LigandPNGBDBM7245((3Z)-5-fluoro-3-({4-oxo-2H,4H,6H,7H-pyrano[3,4-c]p...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:For the assay, purified cdk/cyclin was added to polystyrene 96-well plates that were precoated with GST-Rb substrate in the presence of ATP. After i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2006
Entry Details Article
PubMed
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